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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T62086 | Tuberculosis inhibitor 5 | ||
Tuberculosis inhibitor 5 (Compound 11i) is a potent anti-tuberculosis agent with no apparent cytotoxicity. tuberculosis inhibitor 5 is an antimycobacterial biphenyl analogue. | |||
T9734 | InhA-IN-2 | CDK | |
InhA-IN-2 directly inhibits InhA and does not require activation by the catalase peroxidase KatG. | |||
T0509 | Cloxiquine | 5-Chloro-8-quinolinol,Dermofungin,Dermofongin | Antibacterial , Antibiotic , PPAR , Parasite , Antifungal |
Cloxiquine (Dermofongin) is a monohalogenated 8-hydroxyquinoline with activity against bacteria, fungi, and protozoa. | |||
T3S1612 | Kuwanon G | Moracenin B,Kuwanone G | Phosphatase , Antibacterial , Bombesin Receptor , AChR , AChE , Glucosidase |
1. Kuwanon G (Moracenin B) as dual inhibitors of PTP1B and α-glucosidase enzymes, as well as insulin sensitizers, it may potentially be utilized as an effective treatment for Type II diabetes mellitus. 2. Kuwanon G has a... | |||
T13223 | Tuberculosis inhibitor 1 | Others | |
Tuberculosis inhibitor 1 is a potent and non-cytotoxic inhibitor of trypanosoma brucei growth (EC50: 5 nM). | |||
T61573 | MtTMPK-IN-5 | ||
MtTMPK-IN-5 (compound 17) is a highly effective inhibitor of M. tuberculosis thymidylate kinase (Mtb TMPK), demonstrating remarkable enzyme inhibitory activity with an IC50 value of 34 μM. Additionally, MtTMPK-IN-5 exhib... | |||
TNU1149 | 5’-Azido-5’-deoxythymidine | ||
Nucleoside Derivatives - 5’-Modified nucleosides, Azido-nucleosides; Drugs and Inhibitors; Inhibitor of mycobacterium tuberculosis monophosphate kinase (TMPKmt) | |||
T61796 | MtTMPK-IN-1 | ||
MtTMPK-IN-1 (compound 3) is a highly effective inhibitor of Mycobacterium tuberculosis thymidylate kinase (Mt TMPK), exhibiting an IC50 value of 2.5 μM. It displays moderate to weak activity against Mtb H37Rv while demon... | |||
T62305 | MtTMPK-IN-2 | ||
MtTMPK-IN-2 (compound 15), a potent inhibitor of Mycobacterium tuberculosis thymidylate kinase (Mt TMPK), demonstrates an IC50 value of 1.1 μM. This compound effectively inhibits Mtb H37Rv with a minimum inhibitory conce... | |||
T62897 | MtTMPK-IN-3 | ||
MtTMPK-IN-3 (compound 25) is a potent inhibitor of Mycobacterium tuberculosis thymidylate kinase (MtTMPK) with an IC50 value of 0.12 μM. It also demonstrates inhibitory activity against Mtb H37Rv with a MIC of 12.5 μM an... | |||
T62081 | Mt KARI-IN-5 | ||
Mt KARI-IN-5 (compound 6c) was a potent inhibitor of Mycobacterium tuberculosis ketohydrin reductase I (MtbKARI) (Ki: 4.72 μM). Mt KARI-IN-5 exhibited inhibition of MtbH37Rv activity with a MIC value of 1.56 μM, low cyto... | |||
T62338 | IMPDH2-IN-2 | ||
IMPDH2-IN-2 is a potent inhibitor of inosine 5'-monophosphate dehydrogenase (IMPDH) (Ki,app: 14 μM) and a potential anti-tuberculosis agent. IMPDH2-IN-2 has a moderate antibacterial effect with MIC values of 6.3 and 11 μ... |